Product Name :
RVX-208
CAS :
1044870-39-4
Formula :
C20H22N2O5
MW:
370.4
Description :
Apabetalone (RVX-208) is an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. Apabetalone has C50s are 87±10 ?M and 0.51±0.041 ?M for BD1 and BD2, respectively. Apabetalone binds to the acetyl-lysine binding pocket in a peptide-competitive way, which accounts for its pharmacological activity.
Purity :
98%
Ships Within:
24 Hours
Storage Condition :
-20°C
Shipping :
Ambient Temperature
Availability :
In Stock
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